2026-09-19_00000237
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ligand
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9XHC
Structure of SARS-CoV-2 Mpro complexed with 5bf;
X-ray diffraction 1.80Å
Protein #1
306 residues (99% resolved)
Raw Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Canonical Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Non polymer #2
A1MCK
InChI=1S/C26H30BrClN2O5/c1-33-22-11-16(12-23(34-2)26(22)35-3)20-14-21(29-10-6-4-5-7-24(29)31)18-13-17(27)8-9-19(18)30(20)25(32)15-28/h8-9,11-13,20-21H,4-7,10,14-15H2,1-3H3/t20-,21-/m0/s1
InChI=1S/C26H30BrClN2O5/c1-33-22-11-16(12-23(34-2)26(22)35-3)20-14-21(29-10-6-4-5-7-24(29)31)18-13-17(27)8-9-19(18)30(20)25(32)15-28/h8-9,11-13,20-21H,4-7,10,14-15H2,1-3H3/t20-,21-/m0/s1
SMILES: COc1cc(cc(c1OC)OC)[C@@H]2C[C@@H](c3cc(ccc3N2C(=O)CCl)Br)N4CCCCCC4=O
COc1cc(cc(c1OC)OC)[C@@H]2C[C@@H](c3cc(ccc3N2C(=O)CCl)Br)N4CCCCCC4=O
Non polymer #3
DMS
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
SMILES: CS(=O)C
CS(=O)C
Biounit #1
homo-dimer
Download coordinates
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Model
Reference
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