2026-09-12_00000342|ligand|9ZU3

Crystal structure of BRD9 bromodomain bound to BZ1; X-ray diffraction 1.15Å
Protein #1 129 residues (82% resolved)

MGSSHHHHHHHHHSSGENLYFQGAENESTPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSK

MGSSHHHHHHHHHSSGENLYFQGAENESTPIQQLLEHFLRQLQRKDPHGFFAFPVTDAIAPGYSMIIKHPMDFGTMKDKIVANEYKSVTEFKADFKLMCDNAMTYNRPDTVYYKLAKKILHAGFKMMSK
Non polymer #2 A1C4C

InChI=1S/C13H15ClN4O/c1-18-13(19)12(14)11(8-16-18)17-10-4-2-9(3-5-10)6-7-15/h2-5,8,17H,6-7,15H2,1H3

CN1C(=O)C(=C(C=N1)Nc2ccc(cc2)CCN)Cl
Download coordinates
Reference