2026-09-05_00000187
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ligand
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9Q9X
Redesigned nitrobindin to bind fluorescent ligand;
X-ray diffraction 1.78Å
Protein #1
187 residues (86% resolved)
Raw Sequence ...
GSSHHHHHHSSGENLYFQGSHMIQLQQLQNPGESPPVHPFVAPLSYLLGTWRGQGEGEYPTIPSFRYGEEIRFSHSGKPVIAYTQKTWKLESGAPMTAMSGYFRPRPDGSIEVVVTASHGAVAVFKGTYNVDEQSIKLKSDLVGNSSFMKEISAEFELVDGKLSYVVRMSTTTNPLQPLAKAILDKL
Canonical Sequence ...
GSSHHHHHHSSGENLYFQGSHMIQLQQLQNPGESPPVHPFVAPLSYLLGTWRGQGEGEYPTIPSFRYGEEIRFSHSGKPVIAYTQKTWKLESGAPMTAMSGYFRPRPDGSIEVVVTASHGAVAVFKGTYNVDEQSIKLKSDLVGNSSFMKEISAEFELVDGKLSYVVRMSTTTNPLQPLAKAILDKL
Non polymer #2
A1I5B
InChI=1S/C28H31N5O5/c1-8-9-29-20(34)12-32-25(35)16-10-19(31-14(4)5)24-22-17(26(36)33(15(6)7)28(24)38)11-18(30-13(2)3)23(21(16)22)27(32)37/h1,10-11,13-15,30-31H,9,12H2,2-7H3,(H,29,34)
InChI=1S/C28H31N5O5/c1-8-9-29-20(34)12-32-25(35)16-10-19(31-14(4)5)24-22-17(26(36)33(15(6)7)28(24)38)11-18(30-13(2)3)23(21(16)22)27(32)37/h1,10-11,13-15,30-31H,9,12H2,2-7H3,(H,29,34)
SMILES: CC(C)Nc1cc2c3c4c1C(=O)N(C(=O)c4cc(c3C(=O)N(C2=O)CC(=O)NCC#C)NC(C)C)C(C)C
CC(C)Nc1cc2c3c4c1C(=O)N(C(=O)c4cc(c3C(=O)N(C2=O)CC(=O)NCC#C)NC(C)C)C(C)C
Non polymer #3
NA
InChI=1S/Na/q+1
InChI=1S/Na/q+1
SMILES: [Na+]
[Na+]
Biounit #1
homo-dimer
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Model
Reference
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