2026-09-05_00000086|ligand|29US

KAT6A SURFACE MUTANT IN COMPLEX WITH QUINOLINE INHIBITOR COMPOUND-1; X-ray diffraction 2.70Å
Protein #1 272 residues (99% resolved)

GSPSVIEFGKYEIHTWYSSPYPQEYSRLPKLYLCEFCLKYMKSRTILQQHMKKCGWFHPPANEIYRKNNISVFEVDGNVSTIYCQNLCLLAKLFLDH(ALY)TLYYDVEPFLFYVLTQNDVKGCHLVGYFSKEKHSQQKYNVSSIMILPQYQRKGYGRFLIDFSYLLSKREGQAGSPEKPLSDLGRLSYMAYWKSVILECLYHQNDKQISIKKLSKLTGISPQDITSTLHHLRMLDFRSDQFVIIRREKLIQDHMAKLQLNLRPVDVDPESLRWTP

GSPSVIEFGKYEIHTWYSSPYPQEYSRLPKLYLCEFCLKYMKSRTILQQHMKKCGWFHPPANEIYRKNNISVFEVDGNVSTIYCQNLCLLAKLFLDHKTLYYDVEPFLFYVLTQNDVKGCHLVGYFSKEKHSQQKYNVSSIMILPQYQRKGYGRFLIDFSYLLSKREGQAGSPEKPLSDLGRLSYMAYWKSVILECLYHQNDKQISIKKLSKLTGISPQDITSTLHHLRMLDFRSDQFVIIRREKLIQDHMAKLQLNLRPVDVDPESLRWTP
Non polymer #2 A1J4W

InChI=1S/C21H19N3O4S/c1-13-7-8-14-5-4-6-19(20(14)22-13)29(26,27)23-21(25)18-11-15-9-10-16(24(2)3)12-17(15)28-18/h4-12H,1-3H3,(H,23,25)

Cc1ccc2cccc(c2n1)S(=O)(=O)NC(=O)c3cc4ccc(cc4o3)N(C)C
Non polymer #3 ZN

InChI=1S/Zn/q+2

[Zn+2]
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Reference