2026-08-08_00000066|ligand|25HR

Cryo-EM structure of Pseudomonas aeruginosa FtsQBLWI in complex with imipenem; Electron microscopy 3.60Å
Protein #1 287 residues (68% resolved)

MNGVLLRHQQPGGLGRAPRKPMPRGASRLVAKEPLSVRLPKADFSFLKYLAWPLLLAVLGYGAYRGAEYILPYADRPIAKVSVEGDLSYISQRAVQQRISPYLAASFFTIDLAGMRGQLEQMPWIAHAEVRRVWPDQVVIRLDEQLPIARWGDEALLNNQGQAFTPKELANYEHLPRLHGPQRAQQQVMQQYQLLSQLLRPLGFSIARLEMSDRGGWALTTAQGVEIQIGRDHVVDKIRRFVSIYDKALKDQISNIARIDLRYPNGLAVAWREPVTPATVATASAVQ

MNGVLLRHQQPGGLGRAPRKPMPRGASRLVAKEPLSVRLPKADFSFLKYLAWPLLLAVLGYGAYRGAEYILPYADRPIAKVSVEGDLSYISQRAVQQRISPYLAASFFTIDLAGMRGQLEQMPWIAHAEVRRVWPDQVVIRLDEQLPIARWGDEALLNNQGQAFTPKELANYEHLPRLHGPQRAQQQVMQQYQLLSQLLRPLGFSIARLEMSDRGGWALTTAQGVEIQIGRDHVVDKIRRFVSIYDKALKDQISNIARIDLRYPNGLAVAWREPVTPATVATASAVQ
Protein #2 97 residues (97% resolved)

MSRLFVKRLPTGSFLMLLLYIGLLLSAIAVAYSTYWNRQLLNSLYSELSVRDKAQAEWGRLILEQSTWTAHSRIESLAVEQLRMRVPDPAEVRMVAP

MSRLFVKRLPTGSFLMLLLYIGLLLSAIAVAYSTYWNRQLLNSLYSELSVRDKAQAEWGRLILEQSTWTAHSRIESLAVEQLRMRVPDPAEVRMVAP
Protein #3 94 residues (95% resolved)

MRLRSPYWLFVVLILALAGLQYRLWVGDGSLAQVRDLQKQIADQHGENERLLERNRILEAEVAELKKGTETVEERARHELGMVKDGETLYQLAK

MRLRSPYWLFVVLILALAGLQYRLWVGDGSLAQVRDLQKQIADQHGENERLLERNRILEAEVAELKKGTETVEERARHELGMVKDGETLYQLAK
Protein #4 399 residues (90% resolved)

MLSVLRPFPSPLLSRHGIDLDFPLLAGCLALLGLGLVMVTSASSEVAAAQSGNPLYFSVRHLIYLVIGLISCGLTMMVPMATWQRWGWKLLLVAFGLLVLVITPGIGREVNGSMRWIGFGLFNIQPSEIAKVCVVIFMAGYLIRRQQEVRESWMGFFKPFVVLLPMAGLLLREPDFGATVVMMGAAAAMLFLGGVGLFRFGLMVLLAVGAVVLLIQTQPYRMARLTNFTDPWADQFGAGYQLSQALIAFGRGGWLGMGLGNSIQKQFYLPEAHTDFVFAVLAEELGIVGALATVALFVFVSLRALYIGIWAEQAKQFFSAYVAYGLAFLWIGQFLINIGVNVGLLPTKGLTLPFLSYGGSSLVICCACLGMLLRIEWERRTHLGSEEYEFNEEDFADER

MLSVLRPFPSPLLSRHGIDLDFPLLAGCLALLGLGLVMVTSASSEVAAAQSGNPLYFSVRHLIYLVIGLISCGLTMMVPMATWQRWGWKLLLVAFGLLVLVITPGIGREVNGSMRWIGFGLFNIQPSEIAKVCVVIFMAGYLIRRQQEVRESWMGFFKPFVVLLPMAGLLLREPDFGATVVMMGAAAAMLFLGGVGLFRFGLMVLLAVGAVVLLIQTQPYRMARLTNFTDPWADQFGAGYQLSQALIAFGRGGWLGMGLGNSIQKQFYLPEAHTDFVFAVLAEELGIVGALATVALFVFVSLRALYIGIWAEQAKQFFSAYVAYGLAFLWIGQFLINIGVNVGLLPTKGLTLPFLSYGGSSLVICCACLGMLLRIEWERRTHLGSEEYEFNEEDFADER
Protein #5 579 residues (95% resolved)

MKLNYFQGALYPWRFCVIVGLLLAMVGAIVWRIVDLHVIDHDFLKGQGDARSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKVSVGTKGYRENAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLPTATEQQQVNAAPAKGGRG

MKLNYFQGALYPWRFCVIVGLLLAMVGAIVWRIVDLHVIDHDFLKGQGDARSVRHIAIPAHRGLITDRNGEPLAVSTPVTTLWANPKELMTAKERWPQLAAALGQDTKLFADRIEQNAEREFIYLVRGLTPEQGEGVIALKVPGVYSIEEFRRFYPAGEVVAHAVGFTDVDDRGREGIELAFDEWLAGVPGKRQVLKDRRGRVIKDVQVTKNAKPGKTLALSIDLRLQYLAHRELRNALLENGAKAGSLVIMDVKTGEILAMTNQPTYNPNNRRNLQPAAMRNRAMIDVFEPGSTVKPFSMSAALASGRWKPSDIVDVYPGTLQIGRYTIRDVSRNSRQLDLTGILIKSSNVGISKIAFDIGAESIYSVMQQVGLGQDTGLGFPGERVGNLPNHRKWPKAETATLAYGYGLSVTAIQLAHAYAALANDGKSVPLSMTRVDRVPDGVQVISPEVASTVQGMLQQVVEAQGGVFRAQVPGYHAAGKSGTARKVSVGTKGYRENAYRSLFAGFAPATDPRIAMVVVIDEPSKAGYFGGLVSAPVFSKVMAGALRLMNVPPDNLPTATEQQQVNAAPAKGGRG
Non polymer #6 A1H3N

InChI=1S/C12H19N3O4S/c1-7(17)8(5-16)9-4-10(11(15-9)12(18)19)20-3-2-14-6-13/h5-10,17H,2-4H2,1H3,(H2,13,14)(H,18,19)/t7-,8-,9-,10-/m1/s1

[H]/N=C/NCCS[C@@H]1C[C@@H](N=C1C(=O)O)[C@H](C=O)[C@@H](C)O
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Reference