2026-08-01_00000411|ligand|9YBX

ARID1B ARID bound to compound C-1 (5-fluoro-2-(1H-pyrrolo[2,3-b]pyridine-3-sulfonamido)benzoic acid); X-ray diffraction 1.45Å
Protein #1 120 residues (90% resolved)

GGEKITKVYELGNEPERKLWVDRYLTFMEERGSPVSSLPAVGKKPLDLFRLYVCVKEIGGLAQVNKNKKWRELATNLNVGTSSSAASSLKKQYIQYLFAFECKIERGEEPPPEVFSTGDT

GGEKITKVYELGNEPERKLWVDRYLTFMEERGSPVSSLPAVGKKPLDLFRLYVCVKEIGGLAQVNKNKKWRELATNLNVGTSSSAASSLKKQYIQYLFAFECKIERGEEPPPEVFSTGDT
Non polymer #2 A1CT8

InChI=1S/C14H10FN3O4S/c15-8-3-4-11(10(6-8)14(19)20)18-23(21,22)12-7-17-13-9(12)2-1-5-16-13/h1-7,18H,(H,16,17)(H,19,20)

c1cc2c(c[nH]c2nc1)S(=O)(=O)Nc3ccc(cc3C(=O)O)F
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Reference