2026-08-01_00000212|ligand|32RY

CRYSTAL STRUCTURE OF BRD4-BD1 IN COMPLEX WITH COMPOUND 14; X-ray diffraction 1.92Å
Protein #1 127 residues (98% resolved)

SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE

SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE
Non polymer #2 A1KEY

InChI=1S/C14H15N5/c1-10-3-5-12(6-4-10)8-15-13-7-11(2)17-14-18-16-9-19(13)14/h3-7,9,15H,8H2,1-2H3

Cc1ccc(cc1)CNc2cc(nc3n2cnn3)C
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Reference