2026-08-01_00000210|ligand|32PP

CRYSTAL STRUCTURE OF BRD4 BD1 IN COMPLEX WITH Compound 9; X-ray diffraction 1.44Å
Protein #1 127 residues (98% resolved)

SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE

SMNPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEE
Non polymer #2 A1KEP

InChI=1S/C14H16N6/c1-10-8-13(18-20-11(2)16-17-14(10)20)19(3)9-12-6-4-5-7-15-12/h4-8H,9H2,1-3H3

Cc1cc(nn2c1nnc2C)N(C)Cc3ccccn3
Non polymer #3 EDO

InChI=1S/C2H6O2/c3-1-2-4/h3-4H,1-2H2

C(CO)O
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Reference