2026-06-06_00000299|ligand|9YSP

Human DCTPP1 bound to a Class III inhibitor; X-ray diffraction 1.75Å
Protein #1 110 residues (97% resolved)

GRFSFSPEPTLEDIRRLHAEFAAERDWEQFHQPRNLLLALVGEVGELAELFQWKTDGEPGPQGWSPRERAALQEELSDVLIYLVALAARCRVDLPLAVLSKMDINRRRYP

GRFSFSPEPTLEDIRRLHAEFAAERDWEQFHQPRNLLLALVGEVGELAELFQWKTDGEPGPQGWSPRERAALQEELSDVLIYLVALAARCRVDLPLAVLSKMDINRRRYP
Non polymer #2 A1C0C

InChI=1S/C18H20ClN5OS/c1-26-18-21-16(13-2-4-14(19)5-3-13)15(12-20)17(22-18)24-8-6-23(7-9-24)10-11-25/h2-5,25H,6-11H2,1H3

CSc1nc(c(c(n1)N2CCN(CC2)CCO)C#N)c3ccc(cc3)Cl
Non polymer #3 MG

InChI=1S/Mg/q+2

[Mg+2]
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Reference