2026-06-06_00000018|ligand|13LW

Structure of PKMYT1 bound to inhibitor P32-(S); X-ray diffraction 1.95Å
Protein #1 293 residues (97% resolved)

GPGSMHQLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQP

GPGSMHQLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQP
Non polymer #2 A1DG6

InChI=1S/C17H19N3O2/c21-13-7-3-4-11(8-13)14-9-16(22)19-17-15(14)10-18-20(17)12-5-1-2-6-12/h3-4,7-8,10,12,14,21H,1-2,5-6,9H2,(H,19,22)/t14-/m0/s1

c1cc(cc(c1)O)[C@@H]2CC(=O)Nc3c2cnn3C4CCCC4
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Reference