2026-06-06_00000000|ligand|10BT

X-ray Crystal Structure of A High-Affinity Monoclonal Antibody Sequesters Xylazine; X-ray diffraction 1.99Å
Protein #1 234 residues (95% resolved)

EVKLEESGGGLVQPGGSMRLSCVASGFTFSNYWMNWVRQSPEKGLEWVAEIRLKSNNYATHYAESVKGRFTISRDDSTSSGYLQMNNLRTEDTGIHYCTLTLITDYDVMEYWGQGTSVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHHHHHH

EVKLEESGGGLVQPGGSMRLSCVASGFTFSNYWMNWVRQSPEKGLEWVAEIRLKSNNYATHYAESVKGRFTISRDDSTSSGYLQMNNLRTEDTGIHYCTLTLITDYDVMEYWGQGTSVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHHHHHH
Protein #2 215 residues (100% resolved)

DIQMTQSPSSLSASLGGKVTITCKANQDINKYIAWYQHKPGQGPRLLIHYASALQPGIPSRFSGSGSGRDYSFSISNLEPEDIATYYCLQYDNLYTFGGGTKLEIKRARTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC

DIQMTQSPSSLSASLGGKVTITCKANQDINKYIAWYQHKPGQGPRLLIHYASALQPGIPSRFSGSGSGRDYSFSISNLEPEDIATYYCLQYDNLYTFGGGTKLEIKRARTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC
Non polymer #3 A1C4R

InChI=1S/C12H16N2S/c1-9-5-3-6-10(2)11(9)14-12-13-7-4-8-15-12/h3,5-6H,4,7-8H2,1-2H3,(H,13,14)

Cc1cccc(c1NC2=NCCCS2)C
Non polymer #4 CL

InChI=1S/ClH/h1H/p-1

[Cl-]
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Reference