2026-04-25_00000284|ligand|9WQ1

Crystal structure of CNOT6L and YL-333P complex; X-ray diffraction 2.09Å
Protein #1 398 residues (85% resolved)

MLDNLAVHPEQLPPRPWITLKERDQILPSASFTVMCYNVLCDKYATRQLYGYCPSWALNWEYRKKGIMEEIVNCDADIISLQEVETEQYFTLFLPALKERGYDGFFSPKSRAKIMSEQERKHVDGCAIFFKTEKFTLVQKHTVEFNQVAMANSDGSEAMLNRVMTKDNIGVAVVLEVHKELFGAGMKPIHAADKQLLIVANAHMHWDPEYSDVKLIQTMMFVSEVKNILEKASSRPGSPTADPNSIPLVLCADLNSLPDSGVVEYLSNGGVADNHKDFKELRYNECLMNFSCNGKNGSSEGRITHGFQLKSAYENNLMPYTNYTFDFKGVIDYIFYSKTHMNVLGVLGPLDPQWLVENNITGCPHPHIPSDHFSLLTQLELHPPLLPLVNGVHLPNRR

MLDNLAVHPEQLPPRPWITLKERDQILPSASFTVMCYNVLCDKYATRQLYGYCPSWALNWEYRKKGIMEEIVNCDADIISLQEVETEQYFTLFLPALKERGYDGFFSPKSRAKIMSEQERKHVDGCAIFFKTEKFTLVQKHTVEFNQVAMANSDGSEAMLNRVMTKDNIGVAVVLEVHKELFGAGMKPIHAADKQLLIVANAHMHWDPEYSDVKLIQTMMFVSEVKNILEKASSRPGSPTADPNSIPLVLCADLNSLPDSGVVEYLSNGGVADNHKDFKELRYNECLMNFSCNGKNGSSEGRITHGFQLKSAYENNLMPYTNYTFDFKGVIDYIFYSKTHMNVLGVLGPLDPQWLVENNITGCPHPHIPSDHFSLLTQLELHPPLLPLVNGVHLPNRR
Non polymer #2 A1EX4

InChI=1S/C27H26F2N6O/c28-26(29)35-10-7-21-23(32-16-33-24(21)35)34-11-8-27(30,9-12-34)14-17-1-3-18(4-2-17)19-5-6-20-15-31-25(36)22(20)13-19/h1-7,10,13,16,26H,8-9,11-12,14-15,30H2,(H,31,36)

c1cc(ccc1CC2(CCN(CC2)c3c4ccn(c4ncn3)C(F)F)N)c5ccc6c(c5)C(=O)NC6
Non polymer #3 MG

InChI=1S/Mg/q+2

[Mg+2]
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Reference