2026-04-25_00000072|ligand|9K8Y

Structure of PfENT1(T144C,K375C,N60R,Q266R) with inosine- outward-facing state; Electron microscopy 3.76Å
Protein #1 376 residues (96% resolved)

SSKQHFMLSLTFILIGLSSLNVWNTALGLRINFKYNTFQITGLVCSSIVALFVEIPKIMLPFLLGGLSILCAGFQISHSFFTDTQFDTYCLVAFIVIGVVAGLAQTIAFNIGSCMEDNMGGYMSAGIGISGVFIFVINLLLDQFVSPEKHYGVNKAKLLALYIICELCLILAIVFCVCNLDLTNKNNKKDEENKENNATLSYMELFKDSYKAILTMFLVNWLTLQLFPGVGHKKWRESHNISDYNVTIIVGMFQVFDFLSRYPPNLTHIKIFKNFTFSLNKLLVANSLRLLFIPWFILNACVDHPFFKNIVQQCVCMAMLAFTNGWFNTVPFLVFVKELKKAKKCKEIEIISTFLVIAMFVGLFCGIWTTYIYNLF

SSKQHFMLSLTFILIGLSSLNVWNTALGLRINFKYNTFQITGLVCSSIVALFVEIPKIMLPFLLGGLSILCAGFQISHSFFTDTQFDTYCLVAFIVIGVVAGLAQTIAFNIGSCMEDNMGGYMSAGIGISGVFIFVINLLLDQFVSPEKHYGVNKAKLLALYIICELCLILAIVFCVCNLDLTNKNNKKDEENKENNATLSYMELFKDSYKAILTMFLVNWLTLQLFPGVGHKKWRESHNISDYNVTIIVGMFQVFDFLSRYPPNLTHIKIFKNFTFSLNKLLVANSLRLLFIPWFILNACVDHPFFKNIVQQCVCMAMLAFTNGWFNTVPFLVFVKELKKAKKCKEIEIISTFLVIAMFVGLFCGIWTTYIYNLF
Non polymer #2 NOS

InChI=1S/C10H12N4O5/c15-1-4-6(16)7(17)10(19-4)14-3-13-5-8(14)11-2-12-9(5)18/h2-4,6-7,10,15-17H,1H2,(H,11,12,18)/t4-,6-,7-,10-/m1/s1

c1nc2c(n1[C@H]3[C@@H]([C@@H]([C@H](O3)CO)O)O)N=CNC2=O
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Reference