2026-03-21_00000030
|
ligand
|
22DR
Crystal structure of SARS-CoV-2 3CL protease in complex with compound 7c;
X-ray diffraction 1.90Å
Protein #1
308 residues (98% resolved)
Raw Sequence ...
GSSGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Canonical Sequence ...
GSSGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Non polymer #2
A1MDL
InChI=1S/C23H21F4N7O3/c1-31-11-28-17(30-31)10-34-22(35)19-16(7-18(29-21(19)37-2)32-4-3-13(24)9-32)33(23(34)36)8-12-5-14(25)20(27)15(26)6-12/h5-7,11,13H,3-4,8-10H2,1-2H3/t13-/m1/s1
InChI=1S/C23H21F4N7O3/c1-31-11-28-17(30-31)10-34-22(35)19-16(7-18(29-21(19)37-2)32-4-3-13(24)9-32)33(23(34)36)8-12-5-14(25)20(27)15(26)6-12/h5-7,11,13H,3-4,8-10H2,1-2H3/t13-/m1/s1
SMILES: Cn1cnc(n1)CN2C(=O)c3c(cc(nc3OC)N4CC[C@H](C4)F)N(C2=O)Cc5cc(c(c(c5)F)F)F
Cn1cnc(n1)CN2C(=O)c3c(cc(nc3OC)N4CC[C@H](C4)F)N(C2=O)Cc5cc(c(c(c5)F)F)F
Non polymer #3
EDO
InChI=1S/C2H6O2/c3-1-2-4/h3-4H,1-2H2
InChI=1S/C2H6O2/c3-1-2-4/h3-4H,1-2H2
SMILES: C(CO)O
C(CO)O
Biounit #1
homo-dimer
Download coordinates
Tube
Model
Reference
100%