2026-02-07_00000104
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ligand
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9O21
Heparanase P6 in complex with fragment J34;
X-ray diffraction 1.82Å
Protein #1
383 residues (100% resolved)
Raw Sequence ...
KNSTYSRSSVDVLYTFAKCSGLDLIFGLNALLRTSDGQWNSSNAQLLLDYCASKGYNIDWELGNEPNSFRKKAGIFINGSQLGKDFIHLHKLLRKSTFKNAKLYGPDVGQPRGKTAKMLKSFLKAGGEVIDAVTWHHYYLNGRTATLEDFLNPDVLDTFISQVQKVLQVVESTRPGKKVWLGETSSAYGGGAPGLSDTFAAGFMWLDKLGLSARMGIEVVMRQVFFGAGNYHLVDENFDPLPDYWLSLLFKKLVGTKVLMASVQGQDRRKLRVYLHCTNTDNPRYKEGDLTLYAINLHNVTKYLRLPYPFSNKQVDQYLLRPHGPDGLLSKSVQLNGQTLKMVDDQTLPPLKPKPLRPGSSLGLPAFSYAFFVIRNAKVPACI
Canonical Sequence ...
KNSTYSRSSVDVLYTFAKCSGLDLIFGLNALLRTSDGQWNSSNAQLLLDYCASKGYNIDWELGNEPNSFRKKAGIFINGSQLGKDFIHLHKLLRKSTFKNAKLYGPDVGQPRGKTAKMLKSFLKAGGEVIDAVTWHHYYLNGRTATLEDFLNPDVLDTFISQVQKVLQVVESTRPGKKVWLGETSSAYGGGAPGLSDTFAAGFMWLDKLGLSARMGIEVVMRQVFFGAGNYHLVDENFDPLPDYWLSLLFKKLVGTKVLMASVQGQDRRKLRVYLHCTNTDNPRYKEGDLTLYAINLHNVTKYLRLPYPFSNKQVDQYLLRPHGPDGLLSKSVQLNGQTLKMVDDQTLPPLKPKPLRPGSSLGLPAFSYAFFVIRNAKVPACI
Protein #2
74 residues (100% resolved)
Raw Sequence ...
QDVVDLDFFTQEPLHLVSPSFLSVTIDANLATDPRFLILLGSPKLRTLARGLSPAYLRFGGTKTDFLIFDPKKE
Canonical Sequence ...
QDVVDLDFFTQEPLHLVSPSFLSVTIDANLATDPRFLILLGSPKLRTLARGLSPAYLRFGGTKTDFLIFDPKKE
Non polymer #3
A1B72
InChI=1S/C17H22N2O/c1-13(19-10-6-2-3-7-11-19)17(20)15-12-18-16-9-5-4-8-14(15)16/h4-5,8-9,12-13,18H,2-3,6-7,10-11H2,1H3/t13-/m0/s1
InChI=1S/C17H22N2O/c1-13(19-10-6-2-3-7-11-19)17(20)15-12-18-16-9-5-4-8-14(15)16/h4-5,8-9,12-13,18H,2-3,6-7,10-11H2,1H3/t13-/m0/s1
SMILES: C[C@@H](C(=O)c1c[nH]c2c1cccc2)N3CCCCCC3
C[C@@H](C(=O)c1c[nH]c2c1cccc2)N3CCCCCC3
Non polymer #4
ACT
InChI=1S/C2H4O2/c1-2(3)4/h1H3,(H,3,4)/p-1
InChI=1S/C2H4O2/c1-2(3)4/h1H3,(H,3,4)/p-1
SMILES: CC(=O)[O-]
CC(=O)[O-]
Non polymer #5
EDO
InChI=1S/C2H6O2/c3-1-2-4/h3-4H,1-2H2
InChI=1S/C2H6O2/c3-1-2-4/h3-4H,1-2H2
SMILES: C(CO)O
C(CO)O
Non polymer #6
PEG
InChI=1S/C4H10O3/c5-1-3-7-4-2-6/h5-6H,1-4H2
InChI=1S/C4H10O3/c5-1-3-7-4-2-6/h5-6H,1-4H2
SMILES: C(COCCO)O
C(COCCO)O
Biounit #1
hetero-1-1-mer
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Model
Reference
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