2026-01-17_00000394
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ligand
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9XYM
Crystal Structure of SARS-CoV-2 Main Protease (Mpro) in complex with Jun13698;
X-ray diffraction 2.87Å
Protein #1
306 residues (100% resolved)
Raw Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Canonical Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Non polymer #2
A1CR5
InChI=1S/C20H30F3N3O4S/c1-10(2)14(25-18(30)20(21,22)23)17(29)26-8-12-13(19(12,3)4)15(26)16(28)24-11(9-27)6-7-31-5/h9-15H,6-8H2,1-5H3,(H,24,28)(H,25,30)/t11-,12-,13-,14-,15-/m0/s1
InChI=1S/C20H30F3N3O4S/c1-10(2)14(25-18(30)20(21,22)23)17(29)26-8-12-13(19(12,3)4)15(26)16(28)24-11(9-27)6-7-31-5/h9-15H,6-8H2,1-5H3,(H,24,28)(H,25,30)/t11-,12-,13-,14-,15-/m0/s1
SMILES: CC(C)[C@@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](CCSC)C=O)C2(C)C)NC(=O)C(F)(F)F
CC(C)[C@@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](CCSC)C=O)C2(C)C)NC(=O)C(F)(F)F
Biounit #1
homo-dimer
Download coordinates
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Model
Reference
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