2026-01-10_00000377|ligand|9Q1G

Blimp-1 with compound 5; X-ray diffraction 3.70Å
Protein #1 188 residues (85% resolved)

GSKMDMEDADMTLWTEAEFEEKCTYIVNDHPWDSGADGGTSVQAEASLPRNLLFKYATNSEEVIGVMSKEYIPKGTRFGPLIGEIYTNDTVPKNANRKYFWRIYSRGELHHFIDGFNEEKSNWMRYVNPAHSPREQNLAACQNGMNIYFYTIKPIPANQELLVWYCRDFAERLHYPYPGELTMMNLTQ

GSKMDMEDADMTLWTEAEFEEKCTYIVNDHPWDSGADGGTSVQAEASLPRNLLFKYATNSEEVIGVMSKEYIPKGTRFGPLIGEIYTNDTVPKNANRKYFWRIYSRGELHHFIDGFNEEKSNWMRYVNPAHSPREQNLAACQNGMNIYFYTIKPIPANQELLVWYCRDFAERLHYPYPGELTMMNLTQ
Non polymer #2 A1CNQ

InChI=1S/C15H15BrN4O/c16-12-3-1-10(2-4-12)14(15(17)21)20-6-5-11-7-18-9-19-13(11)8-20/h1-4,7,9,14H,5-6,8H2,(H2,17,21)/t14-/m0/s1

c1cc(ccc1[C@@H](C(=O)N)N2CCc3cncnc3C2)Br
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Reference