2026-01-10_00000029|ligand|7I8P

Crystal Structure of 21 bound to CK2a; X-ray diffraction 1.25Å
Protein #1 328 residues (100% resolved)

SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK

SGPVPSRARVYTDVNTHRPSEYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVAAAKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRKEPFFHGHDNYDQLVRIAKVLGTEDLYDYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVK
Non polymer #2 A1BZV

InChI=1S/C33H34ClN5O2/c34-30-19-23(9-11-26(30)24-7-2-1-3-8-24)21-36-15-5-4-14-35-16-6-17-38-32-28-13-18-37-22-29(28)27-12-10-25(33(40)41)20-31(27)39-32/h1-3,7-13,18-20,22,35-36H,4-6,14-17,21H2,(H,38,39)(H,40,41)

c1ccc(cc1)c2ccc(cc2Cl)CNCCCCNCCCNc3c4ccncc4c5ccc(cc5n3)C(=O)O
Non polymer #3 ACT

InChI=1S/C2H4O2/c1-2(3)4/h1H3,(H,3,4)/p-1

CC(=O)[O-]
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Reference