2025-12-20_00000273
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ligand
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9S1O
Crystal structure of DNPH1 bound by compound 18;
X-ray diffraction 1.77Å
Protein #1
152 residues (82% resolved)
Raw Sequence ...
MRPALYFCGSIRGGREDRTLYERIVSRLRRFGTVLTEHVAAAELGARGEEAAGGDRLIHEQDLEWLQQADVVVAEVTQPSLGVGYELGRAVAFNKRILCLFRPQSGRVLSAMIRGAADGSRFQVWDYEEGEVEALLDRYFEADPLEENLYFQ
Canonical Sequence ...
MRPALYFCGSIRGGREDRTLYERIVSRLRRFGTVLTEHVAAAELGARGEEAAGGDRLIHEQDLEWLQQADVVVAEVTQPSLGVGYELGRAVAFNKRILCLFRPQSGRVLSAMIRGAADGSRFQVWDYEEGEVEALLDRYFEADPLEENLYFQ
Non polymer #2
A1JK6
InChI=1S/C27H30N4O2S/c32-26(33)22-7-6-21-8-9-29(16-23(21)11-22)17-24-18-34-27(28-24)31-14-19-10-20(15-31)13-30(12-19)25-4-2-1-3-5-25/h1-7,11,18-20H,8-10,12-17H2,(H,32,33)/t19-,20+
InChI=1S/C27H30N4O2S/c32-26(33)22-7-6-21-8-9-29(16-23(21)11-22)17-24-18-34-27(28-24)31-14-19-10-20(15-31)13-30(12-19)25-4-2-1-3-5-25/h1-7,11,18-20H,8-10,12-17H2,(H,32,33)/t19-,20+
SMILES: c1ccc(cc1)N2C[C@H]3C[C@@H](C2)CN(C3)c4nc(cs4)CN5CCc6ccc(cc6C5)C(=O)O
c1ccc(cc1)N2C[C@H]3C[C@@H](C2)CN(C3)c4nc(cs4)CN5CCc6ccc(cc6C5)C(=O)O
Non polymer #3
CL
InChI=1S/ClH/h1H/p-1
InChI=1S/ClH/h1H/p-1
SMILES: [Cl-]
[Cl-]
Biounit #1
homo-dimer
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Model
Reference
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