2025-12-13_00000111|hard|9M55

Structural insight into determinants of endogenous agonist selectivity of aminergic receptors from octopamine b2 receptor structure; Electron microscopy 3.39Å
Protein #1 402 residues (48% resolved)

MKDHLIHNHHKHEHAHAEHLYFQGSSGSSGMASTLSAEDKAAVERSKMIEKQIQKDKQIYRATHRLLLLGAGESGKNTIVKQMRILHVNGFSEEEKKQKIEDIKKNIRDAILTITGAMSTLVPPVQLQKSENQWRVDYIQDVASSPDFDYPAEFYEHTEILWKDKGVQAAFERSNEYQLIDCAKYFLDRVATIKQLDYTPNEQDILRCRVLTSGIFETKFQVDKVNFHMFDVGAQRDERRKWIQCFNDVTAIIFVTACSSYNMVLREDPNQNRLRASLKLFDSIWNNKWLRDTSVILFLNKQDLLAEKIKAGKSRLEEYFPEFAHYQTPSDAVIETGEDPEVIRAKYFIRDEFLRISTASGDGKHYCYPHFTCSVDTENIRRVFNDCRDIIQRMHLRQYELL

MKDHLIHNHHKHEHAHAEHLYFQGSSGSSGMASTLSAEDKAAVERSKMIEKQIQKDKQIYRATHRLLLLGAGESGKNTIVKQMRILHVNGFSEEEKKQKIEDIKKNIRDAILTITGAMSTLVPPVQLQKSENQWRVDYIQDVASSPDFDYPAEFYEHTEILWKDKGVQAAFERSNEYQLIDCAKYFLDRVATIKQLDYTPNEQDILRCRVLTSGIFETKFQVDKVNFHMFDVGAQRDERRKWIQCFNDVTAIIFVTACSSYNMVLREDPNQNRLRASLKLFDSIWNNKWLRDTSVILFLNKQDLLAEKIKAGKSRLEEYFPEFAHYQTPSDAVIETGEDPEVIRAKYFIRDEFLRISTASGDGKHYCYPHFTCSVDTENIRRVFNDCRDIIQRMHLRQYELL
Protein #2 358 residues (92% resolved)

MDYKDDDDKENLYFQGGSMSELDQLRQEAEQLKNQIRDARKACADATLSQITNNIDPVGRIQMRTRRTLRGHLAKIYAMHWGTDSRLLVSASQDGKLIIWDSYTTNKVHAIPLRSSWVMTCAYAPSGNYVACGGLDNICSIYNLKTREGNVRVSRELAGHTGYLSCCRFLDDNQIVTSSGDTTCALWDIETGQQTTTFTGHTGDVMSLSLAPDTRLFVSGACDASAKLWDVREGMCRQTFTGHESDINAICFFPNGNAFATGSDDATCRLFDLRADQELMTYSHDNIICGITSVSFSKSGRLLLAGYDDFNCNVWDALKADRAGVLAGHDNRVSCLGVTDDGMAVATGSWDSFLKIWN

MDYKDDDDKENLYFQGGSMSELDQLRQEAEQLKNQIRDARKACADATLSQITNNIDPVGRIQMRTRRTLRGHLAKIYAMHWGTDSRLLVSASQDGKLIIWDSYTTNKVHAIPLRSSWVMTCAYAPSGNYVACGGLDNICSIYNLKTREGNVRVSRELAGHTGYLSCCRFLDDNQIVTSSGDTTCALWDIETGQQTTTFTGHTGDVMSLSLAPDTRLFVSGACDASAKLWDVREGMCRQTFTGHESDINAICFFPNGNAFATGSDDATCRLFDLRADQELMTYSHDNIICGITSVSFSKSGRLLLAGYDDFNCNVWDALKADRAGVLAGHDNRVSCLGVTDDGMAVATGSWDSFLKIWN
Protein #3 99 residues (49% resolved)

MSYYHHHHHHDYDIPTTENLYFQGAMGSMASNNTASIAQARKLVEQLKMEANIDRIKVSKAAADLMAYCEAHAKEDPLLTPVPASENPFREKKFFSAIL

MSYYHHHHHHDYDIPTTENLYFQGAMGSMASNNTASIAQARKLVEQLKMEANIDRIKVSKAAADLMAYCEAHAKEDPLLTPVPASENPFREKKFFSAIL
Protein #4 425 residues (64% resolved)

MKTIIALSYIFCLVFADYKDDDDKENLYFQGMTVAAPNASLANLTEEAQADDESWESVLKLVLKTLALVTIISSAVFGNLLVVTSVIRHHKLRITTNYFIVSLALADTLVALFAMTFNASVTISGRWLFNQTVCDFWNSCDVLFSTASIMHLCCISVDRYYAIIKPLEYPTKITGRTVAIMLTCAWVSSGLISFIPIFLGWYTTNEHLVYKVEHPDECIFVVNKPYAIISSSVSFWIPCCIMLFTYWRIYVEATRQEKMLCKSQMGPGMLCRNSTDQSMPNVHAPPHRNSHGDDPESGQSTPTKRTINKMKREHKAAKTLGIIMGAFILCWLPFFLWYVSITMCGDACPCPELVVDLLFWIGYLNSSLNPVIYAYFNREFRQAFKETLQAIFCSSRCSSCATGSRQTGGRPPGRTHHHHHHHHHH

MKTIIALSYIFCLVFADYKDDDDKENLYFQGMTVAAPNASLANLTEEAQADDESWESVLKLVLKTLALVTIISSAVFGNLLVVTSVIRHHKLRITTNYFIVSLALADTLVALFAMTFNASVTISGRWLFNQTVCDFWNSCDVLFSTASIMHLCCISVDRYYAIIKPLEYPTKITGRTVAIMLTCAWVSSGLISFIPIFLGWYTTNEHLVYKVEHPDECIFVVNKPYAIISSSVSFWIPCCIMLFTYWRIYVEATRQEKMLCKSQMGPGMLCRNSTDQSMPNVHAPPHRNSHGDDPESGQSTPTKRTINKMKREHKAAKTLGIIMGAFILCWLPFFLWYVSITMCGDACPCPELVVDLLFWIGYLNSSLNPVIYAYFNREFRQAFKETLQAIFCSSRCSSCATGSRQTGGRPPGRTHHHHHHHHHH
Protein #5 308 residues (75% resolved)

MKDHLIHNHHKHEHAHAEHLYFQGSSGSSGDVQLVESGGGLVQPGGSRKLSCSASGFAFSSFGMHWVRQAPEKGLEWVAYISSGSGTIYYADTVKGRFTISRDDPKNTLFLQMTSLRSEDTAMYYCVRSIYYYGSSPFDFWGQGTTLTVSSGGGGSGGGGSGGGGSDIVMTQATSSVPVTPGESVSISCRSSKSLLHSNGNTYLYWFLQRPGQSPQLLIYRMSNLASGVPDRFSGSGSGTAFTLTISRLEAEDVGVYYCMQHLEYPLTFGAGTKLELKSAWSHPQFEKGGGSGGGSGGSAWSHPQFEK

MKDHLIHNHHKHEHAHAEHLYFQGSSGSSGDVQLVESGGGLVQPGGSRKLSCSASGFAFSSFGMHWVRQAPEKGLEWVAYISSGSGTIYYADTVKGRFTISRDDPKNTLFLQMTSLRSEDTAMYYCVRSIYYYGSSPFDFWGQGTTLTVSSGGGGSGGGGSGGGGSDIVMTQATSSVPVTPGESVSISCRSSKSLLHSNGNTYLYWFLQRPGQSPQLLIYRMSNLASGVPDRFSGSGSGTAFTLTISRLEAEDVGVYYCMQHLEYPLTFGAGTKLELKSAWSHPQFEKGGGSGGGSGGSAWSHPQFEK
Non polymer #6 A1L8N

InChI=1S/C10H14N2/c1-8-4-5-10(9(2)6-8)12-7-11-3/h4-7H,1-3H3,(H,11,12)

Cc1ccc(c(c1)C)/N=C/NC
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Reference