2025-11-08_00000075|hard|9I5E

A Coiled Coil Module Strategy for High-Resolution Cryo-EM Structures of Small Proteins for Drug Discovery; Electron microscopy 3.77Å
Protein #1 204 residues (100% resolved)

MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRLHKELKQLEEELQAIEEQLAQLQWKAQARKEKLAQLKEKL

MTEYKLVVVGACGVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETCLLDILDTAGQEEYSAMRDQYMRTGEGFLCVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKCDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRLHKELKQLEEELQAIEEQLAQLQWKAQARKEKLAQLKEKL
Protein #2 122 residues (100% resolved)

VQLQESGGGLVQAGDSLRLSCAASGRTFSTYPMGWFRQAPGKEREFVAASSSRAYYADSVKGRFTISRNNAKNTVYLQMNSLKPEDTAVYYCVADSSPYYRRYDAAQDYDYWGQGTQVTVSS

VQLQESGGGLVQAGDSLRLSCAASGRTFSTYPMGWFRQAPGKEREFVAASSSRAYYADSVKGRFTISRNNAKNTVYLQMNSLKPEDTAVYYCVADSSPYYRRYDAAQDYDYWGQGTQVTVSS
Non polymer #3 GDP

InChI=1S/C10H15N5O11P2/c11-10-13-7-4(8(18)14-10)12-2-15(7)9-6(17)5(16)3(25-9)1-24-28(22,23)26-27(19,20)21/h2-3,5-6,9,16-17H,1H2,(H,22,23)(H2,19,20,21)(H3,11,13,14,18)/t3-,5-,6-,9-/m1/s1

c1nc2c(n1[C@H]3[C@@H]([C@@H]([C@H](O3)CO[P@](=O)(O)OP(=O)(O)O)O)O)N=C(NC2=O)N
Non polymer #4 M1X

InChI=1S/C32H37ClFN7O2/c1-21(34)31(42)41-17-16-40(18-23(41)11-13-35)30-25-12-15-39(28-10-4-7-22-6-3-9-26(33)29(22)28)19-27(25)36-32(37-30)43-20-24-8-5-14-38(24)2/h3-4,6-7,9-10,21,23-24H,5,8,11-12,14-20H2,1-2H3/t21-,23-,24-/m0/s1

C[C@@H](C(=O)N1CCN(C[C@@H]1CC#N)c2c3c(nc(n2)OC[C@@H]4CCCN4C)CN(CC3)c5cccc6c5c(ccc6)Cl)F
Non polymer #5 MG

InChI=1S/Mg/q+2

[Mg+2]
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Reference