2025-11-01_00000208
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ligand
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9H7R
MITF in complex with 6-((1-hydroxycyclohexyl)ethynyl)-1-phenyl-1H-indole-2-carboxylic acid;
X-ray diffraction 2.52Å
Protein #1
83 residues (93% resolved)
Raw Sequence ...
GAMRFNINDRIKELGTLIPKSNDPDMRWNKGTILKASVDYIRKLQREQQRAKELENRQKKLEHANRHLLLRIQELEMQARAHG
Canonical Sequence ...
GAMRFNINDRIKELGTLIPKSNDPDMRWNKGTILKASVDYIRKLQREQQRAKELENRQKKLEHANRHLLLRIQELEMQARAHG
Non polymer #2
A1IS5
InChI=1S/C23H21NO3/c25-22(26)21-16-18-10-9-17(11-14-23(27)12-5-2-6-13-23)15-20(18)24(21)19-7-3-1-4-8-19/h1,3-4,7-10,15-16,27H,2,5-6,12-13H2,(H,25,26)
InChI=1S/C23H21NO3/c25-22(26)21-16-18-10-9-17(11-14-23(27)12-5-2-6-13-23)15-20(18)24(21)19-7-3-1-4-8-19/h1,3-4,7-10,15-16,27H,2,5-6,12-13H2,(H,25,26)
SMILES: c1ccc(cc1)n2c3cc(ccc3cc2C(=O)O)C#CC4(CCCCC4)O
c1ccc(cc1)n2c3cc(ccc3cc2C(=O)O)C#CC4(CCCCC4)O
Non polymer #3
NA
InChI=1S/Na/q+1
InChI=1S/Na/q+1
SMILES: [Na+]
[Na+]
Non polymer #4
PEG
InChI=1S/C4H10O3/c5-1-3-7-4-2-6/h5-6H,1-4H2
InChI=1S/C4H10O3/c5-1-3-7-4-2-6/h5-6H,1-4H2
SMILES: C(COCCO)O
C(COCCO)O
Biounit #1
homo-trimer
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Model
Reference
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