2025-09-27_00000078|ligand|9GV3

Crystal structure of the complex between Nb474 mutant R53A,D125A and Trypanosoma congolense fructose-1,6-bisphosphate aldolase; X-ray diffraction 1.75Å
Protein #1 387 residues (94% resolved)

MSRRVEVLLTQLPAYNRLKTPYEEELIETAKKMTAPGKGLLAADESTGSCSKRFAGIGLSNTAEHRRQYRALMLECAGFEQYISGVILHDETVYQRASTGETFPQLLRRRGVVPGIKTDCGLEPLVEGADGEQMTAGLDGYVKRAKKYYAVGCRFCKWRNVYKIQNGTVSEAVVRFNAETLARYAVLSQLCGLVPIVEPEVMIDGTHDIETCQRVSQHVWAEVVSALHRHGVVWEGCLLKPNMVVPGAESGQTATAEQVAEYTVKTLARVLPPALPGVTFLSGGLSEVMASEYLNAMNNSPLPRPWKLTFSYARALQSSAIKAWGGKSSGVAAGRRAFMHRAKMNSLAQLGRYNRGDDDKDSQSLYVAGNTYENLYFQSGGHHHHHH

MSRRVEVLLTQLPAYNRLKTPYEEELIETAKKMTAPGKGLLAADESTGSCSKRFAGIGLSNTAEHRRQYRALMLECAGFEQYISGVILHDETVYQRASTGETFPQLLRRRGVVPGIKTDCGLEPLVEGADGEQMTAGLDGYVKRAKKYYAVGCRFCKWRNVYKIQNGTVSEAVVRFNAETLARYAVLSQLCGLVPIVEPEVMIDGTHDIETCQRVSQHVWAEVVSALHRHGVVWEGCLLKPNMVVPGAESGQTATAEQVAEYTVKTLARVLPPALPGVTFLSGGLSEVMASEYLNAMNNSPLPRPWKLTFSYARALQSSAIKAWGGKSSGVAAGRRAFMHRAKMNSLAQLGRYNRGDDDKDSQSLYVAGNTYENLYFQSGGHHHHHH
Protein #2 143 residues (96% resolved)

QVQLQESGGGLVQPGGSLRLSCAASETALTYYAIGWFRQAPGKEREGVSCISAINSGSGARTDYADSVKGRFTISRDDAKNTVTLQMNSLEPEDTARYYCALDTTDRYDSANGRYYCTISSDTYAYWGQGTQVTVSSHHHHHH

QVQLQESGGGLVQPGGSLRLSCAASETALTYYAIGWFRQAPGKEREGVSCISAINSGSGARTDYADSVKGRFTISRDDAKNTVTLQMNSLEPEDTARYYCALDTTDRYDSANGRYYCTISSDTYAYWGQGTQVTVSSHHHHHH
Non polymer #3 ACT

InChI=1S/C2H4O2/c1-2(3)4/h1H3,(H,3,4)/p-1

CC(=O)[O-]
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Reference