2025-09-13_00000189|ligand|9RLO

PARP15 catalytic domain in complex with OUL250; X-ray diffraction 1.90Å
Protein #1 200 residues (99% resolved)

SMNLPEHWTDMNHQLFCMVQLEPGQSEYNTIKDKFTRTCSSYAIEKIERIQNAFLWQSYQVKKRQMDIKNDHKNNERLLFHGTDADSVPYVNQHGFNRSCAGKNAVSYGKGTYFAVDASYSAKDTYSKPDSNGRKHMYVVRVLTGVFTKGRAGLVTPPPKNPHNPTDLFDSVTNNTRSPKLFVVFFDNQAYPEYLITFTA

SMNLPEHWTDMNHQLFCMVQLEPGQSEYNTIKDKFTRTCSSYAIEKIERIQNAFLWQSYQVKKRQMDIKNDHKNNERLLFHGTDADSVPYVNQHGFNRSCAGKNAVSYGKGTYFAVDASYSAKDTYSKPDSNGRKHMYVVRVLTGVFTKGRAGLVTPPPKNPHNPTDLFDSVTNNTRSPKLFVVFFDNQAYPEYLITFTA
Non polymer #2 A1JG9

InChI=1S/C15H11N3O4/c16-13(19)8-1-3-9(4-2-8)22-10-5-6-11-12(7-10)15(21)18-17-14(11)20/h1-7H,(H2,16,19)(H,17,20)(H,18,21)

c1cc(ccc1C(=O)N)Oc2ccc3c(c2)C(=O)NNC3=O
Non polymer #3 DMS

InChI=1S/C2H6OS/c1-4(2)3/h1-2H3

CS(=O)C
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Reference