2025-08-30_00000057
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ligand
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9DE3
Crystal structure of NDM-1 complexed with compound 28;
X-ray diffraction 2.15Å
Protein #1
233 residues (98% resolved)
Raw Sequence ...
GSHMGDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR
Canonical Sequence ...
GSHMGDQRFGDLVFRQLAPNVWQHTSYLDMPGFGAVASNGLIVRDGGRVLVVDTAWTDDQTAQILNWIKQEINLPVALAVVTHAHQDKMGGMDALHAAGIATYANALSNQLAPQEGMVAAQHSLTFAANGWVEPATAPNFGPLKVFYPGPGHTSDNITVGIDGTDIAFGGCLIKDSKAKSLGNLGDADTEHYAASARAFGAAFPKASMIVMSHSAPDSRAAITHTARMADKLR
Non polymer #2
A1A4C
InChI=1S/C21H29N2O4P/c1-15-19(14-28(25,26)27)18-9-8-17(22-10-4-5-11-22)12-20(18)23(21(15)24)13-16-6-2-3-7-16/h8-9,12,16H,2-7,10-11,13-14H2,1H3,(H2,25,26,27)
InChI=1S/C21H29N2O4P/c1-15-19(14-28(25,26)27)18-9-8-17(22-10-4-5-11-22)12-20(18)23(21(15)24)13-16-6-2-3-7-16/h8-9,12,16H,2-7,10-11,13-14H2,1H3,(H2,25,26,27)
SMILES: CC1=C(c2ccc(cc2N(C1=O)CC3CCCC3)N4CCCC4)CP(=O)(O)O
CC1=C(c2ccc(cc2N(C1=O)CC3CCCC3)N4CCCC4)CP(=O)(O)O
Non polymer #3
ZN
InChI=1S/Zn/q+2
InChI=1S/Zn/q+2
SMILES: [Zn+2]
[Zn+2]
Biounit #1
monomer
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Model
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