2025-07-05_00000201|medium|9JF4

cryo-EM structure of Neuromedin B receptor in complex with PD168368; Electron microscopy 3.60Å
Protein #1 520 residues (75% resolved)

DYKDDDAMPSKSLSNLSVTTGANESGSVPEGWERDFLPASDGTTTELVIRCVIPSLYLLIITVGLLGNIMLVKIFITNSAMRSVPNIFISNLAAGDLLLLLTCVPVDASRYFFDEWMFGKVGCKLIPVIQLTSVGVSVWTLTALSADRYRAIVNPMDMQTSGALLRTCVKAMGIWVVSVLLAVPEAVFSEVARISSLDNSSFTACIPYPQTDELHPKIHSVLIFLVYFLIPLAIISIYYYHIAKHLKEKAKAGAEIAAHPDAFLFLLFAAFGVVLTGDPEDRALWAELLALVERAAPGIARALAAAYRAAEEAYRAGGPVAGFRAGILGACAGVDAETRLPLTARIVDLLRTIRALRDDEAALRALVDALGAELRALLAPVAADAEELDALLARLADLALVALRELAKLSESEMDAFIADLTAAVEAMAKQMETRKRLAKIVLVFVGCFIFCWFPNHILYMYRSFNYNEIDPSLGHMIVTLVARVLSFGNSCVNPFALYLLSESFRRHFNSQLCHHHHHH

DYKDDDAMPSKSLSNLSVTTGANESGSVPEGWERDFLPASDGTTTELVIRCVIPSLYLLIITVGLLGNIMLVKIFITNSAMRSVPNIFISNLAAGDLLLLLTCVPVDASRYFFDEWMFGKVGCKLIPVIQLTSVGVSVWTLTALSADRYRAIVNPMDMQTSGALLRTCVKAMGIWVVSVLLAVPEAVFSEVARISSLDNSSFTACIPYPQTDELHPKIHSVLIFLVYFLIPLAIISIYYYHIAKHLKEKAKAGAEIAAHPDAFLFLLFAAFGVVLTGDPEDRALWAELLALVERAAPGIARALAAAYRAAEEAYRAGGPVAGFRAGILGACAGVDAETRLPLTARIVDLLRTIRALRDDEAALRALVDALGAELRALLAPVAADAEELDALLARLADLALVALRELAKLSESEMDAFIADLTAAVEAMAKQMETRKRLAKIVLVFVGCFIFCWFPNHILYMYRSFNYNEIDPSLGHMIVTLVARVLSFGNSCVNPFALYLLSESFRRHFNSQLCHHHHHH
Non polymer #2 A1D63

InChI=1S/C31H34N6O4/c1-30(19-22-20-33-26-10-4-3-9-25(22)26,36-29(39)35-23-12-14-24(15-13-23)37(40)41)28(38)34-21-31(16-6-2-7-17-31)27-11-5-8-18-32-27/h3-5,8-15,18,20,33H,2,6-7,16-17,19,21H2,1H3,(H,34,38)(H2,35,36,39)/t30-/m0/s1

C[C@](Cc1c[nH]c2c1cccc2)(C(=O)NCC3(CCCCC3)c4ccccn4)NC(=O)Nc5ccc(cc5)[N+](=O)[O-]
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Reference