2025-07-05_00000091
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ligand
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9F0T
Structure of KPC-2 complexed with benzoxaborole AK-110;
X-ray diffraction 0.98Å
Protein #1
290 residues (93% resolved)
Raw Sequence ...
MGSSHHHHHHSSGLVPRGSHMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNGQ
Canonical Sequence ...
MGSSHHHHHHSSGLVPRGSHMLTNLVAEPFAKLEQDFGGSIGVYAMDTGSGATVSYRAEERFPLCSSFKGFLAAAVLARSQQQAGLLDTPIRYGKNALVPWSPISEKYLTTGMTVAELSAAAVQYSDNAAANLLLKELGGPAGLTAFMRSIGDTTFRLDRWELELNSAIPGDARDTSSPRAVTESLQKLTLGSALAAPQRQQFVDWLKGNTTGNHRIRAAVPADWAVGDKTGTCGVYGTANDYAVVWPTGRAPIVLAVYTRAPNKDDKHSEAVIAAAARLALEGLGVNGQ
Non polymer #2
A1H8S
InChI=1S/C12H17BN2O4S/c16-13-11-6-2-1-5-10(11)12(19-13)9-14-20(17,18)15-7-3-4-8-15/h1-2,5-6,12,14,16H,3-4,7-9H2/t12-/m1/s1
InChI=1S/C12H17BN2O4S/c16-13-11-6-2-1-5-10(11)12(19-13)9-14-20(17,18)15-7-3-4-8-15/h1-2,5-6,12,14,16H,3-4,7-9H2/t12-/m1/s1
SMILES: B1(c2ccccc2[C@H](O1)CNS(=O)(=O)N3CCCC3)O
B1(c2ccccc2[C@H](O1)CNS(=O)(=O)N3CCCC3)O
Non polymer #3
NA
InChI=1S/Na/q+1
InChI=1S/Na/q+1
SMILES: [Na+]
[Na+]
Biounit #1
monomer
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Model
Reference
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