2025-06-07_00000066
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ligand
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7HE5
PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with AVI-0003659;
X-ray diffraction 1.02Å
Protein #1
169 residues (100% resolved)
Raw Sequence ...
SMVNSFSGYLKLTDNVYIKNADIVEEAKKVKPTVVVNAANVYLKHGGGVAGALNKATNNAMQVESDDYIATNGPLKVGGSCVLSGHNLAKHCLHVVGPNVNKGEDIQLLKSAYENFNQHEVLLAPLLSAGIFGADPIHSLRVCVDTVRTNVYLAVFDKNLYDKLVSSFL
Canonical Sequence ...
SMVNSFSGYLKLTDNVYIKNADIVEEAKKVKPTVVVNAANVYLKHGGGVAGALNKATNNAMQVESDDYIATNGPLKVGGSCVLSGHNLAKHCLHVVGPNVNKGEDIQLLKSAYENFNQHEVLLAPLLSAGIFGADPIHSLRVCVDTVRTNVYLAVFDKNLYDKLVSSFL
Non polymer #2
A1A9H
InChI=1S/C12H12N4O2/c17-6-9(10-2-1-5-18-10)16-12-8-3-4-13-11(8)14-7-15-12/h1-5,7,9,17H,6H2,(H2,13,14,15,16)/t9-/m1/s1
InChI=1S/C12H12N4O2/c17-6-9(10-2-1-5-18-10)16-12-8-3-4-13-11(8)14-7-15-12/h1-5,7,9,17H,6H2,(H2,13,14,15,16)/t9-/m1/s1
SMILES: c1cc(oc1)[C@@H](CO)Nc2c3cc[nH]c3ncn2
c1cc(oc1)[C@@H](CO)Nc2c3cc[nH]c3ncn2
Non polymer #3
CL
InChI=1S/ClH/h1H/p-1
InChI=1S/ClH/h1H/p-1
SMILES: [Cl-]
[Cl-]
Non polymer #4
TFA
InChI=1S/C2HF3O2/c3-2(4,5)1(6)7/h(H,6,7)
InChI=1S/C2HF3O2/c3-2(4,5)1(6)7/h(H,6,7)
SMILES: C(=O)(C(F)(F)F)O
C(=O)(C(F)(F)F)O
Biounit #1
monomer
Download coordinates
Biounit #2
monomer
Download coordinates
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Model
Reference
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