2025-06-07_00000062
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ligand
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7HE1
PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with AVI-0003655;
X-ray diffraction 1.04Å
Protein #1
169 residues (100% resolved)
Raw Sequence ...
SMVNSFSGYLKLTDNVYIKNADIVEEAKKVKPTVVVNAANVYLKHGGGVAGALNKATNNAMQVESDDYIATNGPLKVGGSCVLSGHNLAKHCLHVVGPNVNKGEDIQLLKSAYENFNQHEVLLAPLLSAGIFGADPIHSLRVCVDTVRTNVYLAVFDKNLYDKLVSSFL
Canonical Sequence ...
SMVNSFSGYLKLTDNVYIKNADIVEEAKKVKPTVVVNAANVYLKHGGGVAGALNKATNNAMQVESDDYIATNGPLKVGGSCVLSGHNLAKHCLHVVGPNVNKGEDIQLLKSAYENFNQHEVLLAPLLSAGIFGADPIHSLRVCVDTVRTNVYLAVFDKNLYDKLVSSFL
Non polymer #2
A1A9D
InChI=1S/C12H16N4O/c1-8-3-5-16(10(8)6-17)12-9-2-4-13-11(9)14-7-15-12/h2,4,7-8,10,17H,3,5-6H2,1H3,(H,13,14,15)/t8-,10+/m0/s1
InChI=1S/C12H16N4O/c1-8-3-5-16(10(8)6-17)12-9-2-4-13-11(9)14-7-15-12/h2,4,7-8,10,17H,3,5-6H2,1H3,(H,13,14,15)/t8-,10+/m0/s1
SMILES: C[C@H]1CCN([C@@H]1CO)c2c3cc[nH]c3ncn2
C[C@H]1CCN([C@@H]1CO)c2c3cc[nH]c3ncn2
Non polymer #3
TFA
InChI=1S/C2HF3O2/c3-2(4,5)1(6)7/h(H,6,7)
InChI=1S/C2HF3O2/c3-2(4,5)1(6)7/h(H,6,7)
SMILES: C(=O)(C(F)(F)F)O
C(=O)(C(F)(F)F)O
Biounit #1
monomer
Download coordinates
Biounit #2
monomer
Download coordinates
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Model
Reference
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