2025-05-10_00000136
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ligand
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9BSO
Structure of the SARS-CoV-2 main protease in complex with inhibitor SR-B-13;
X-ray diffraction 1.70Å
Protein #1
306 residues (100% resolved)
Raw Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Canonical Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Non polymer #2
A1ARW
InChI=1S/C20H16Cl2N2OS/c21-16-5-1-3-14(9-16)15-4-2-6-18(10-15)24(20(25)7-8-26)19-11-17(22)12-23-13-19/h1-6,9-13,26H,7-8H2
InChI=1S/C20H16Cl2N2OS/c21-16-5-1-3-14(9-16)15-4-2-6-18(10-15)24(20(25)7-8-26)19-11-17(22)12-23-13-19/h1-6,9-13,26H,7-8H2
SMILES: c1cc(cc(c1)N(c2cc(cnc2)Cl)C(=O)CCS)c3cccc(c3)Cl
c1cc(cc(c1)N(c2cc(cnc2)Cl)C(=O)CCS)c3cccc(c3)Cl
Biounit #1
homo-dimer
Download coordinates
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Model
Reference
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