2025-05-10_00000131
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ligand
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9BSA
Structure of the SARS-CoV-2 main protease in complex with inhibitor VB-B-112;
X-ray diffraction 1.70Å
Protein #1
306 residues (100% resolved)
Raw Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Canonical Sequence ...
SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
Non polymer #2
A1AR5
InChI=1S/C13H9Cl3N2O/c14-9-6-11(8-17-7-9)18(13(19)12(15)16)10-4-2-1-3-5-10/h1-8,12H
InChI=1S/C13H9Cl3N2O/c14-9-6-11(8-17-7-9)18(13(19)12(15)16)10-4-2-1-3-5-10/h1-8,12H
SMILES: c1ccc(cc1)N(c2cc(cnc2)Cl)C(=O)C(Cl)Cl
c1ccc(cc1)N(c2cc(cnc2)Cl)C(=O)C(Cl)Cl
Biounit #1
homo-dimer
Download coordinates
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Model
Reference
100%