2025-04-26_00000164
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ligand
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9DU4
SARS-CoV-2 Mpro in complex with compound 3;
X-ray diffraction 2.42Å
Protein #1
315 residues (96% resolved)
Raw Sequence ...
MSGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQLEHHHHHH
Canonical Sequence ...
MSGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQLEHHHHHH
Non polymer #2
A1BCW
InChI=1S/C21H29N3O6S/c1-30-19-5-3-4-16-15(19)11-18(23-16)21(27)24-17(10-13-6-7-13)20(26)22-14(12-25)8-9-31(2,28)29/h3-5,11,13-14,17,23,25H,6-10,12H2,1-2H3,(H,22,26)(H,24,27)/t14-,17+/m1/s1
InChI=1S/C21H29N3O6S/c1-30-19-5-3-4-16-15(19)11-18(23-16)21(27)24-17(10-13-6-7-13)20(26)22-14(12-25)8-9-31(2,28)29/h3-5,11,13-14,17,23,25H,6-10,12H2,1-2H3,(H,22,26)(H,24,27)/t14-,17+/m1/s1
SMILES: COc1cccc2c1cc([nH]2)C(=O)N[C@@H](CC3CC3)C(=O)N[C@@H](CCS(=O)(=O)C)CO
COc1cccc2c1cc([nH]2)C(=O)N[C@@H](CC3CC3)C(=O)N[C@@H](CCS(=O)(=O)C)CO
Biounit #1
homo-dimer
Download coordinates
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Model
Reference
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