2025-03-29_00000482|ligand|9N2M

Crystal Structure of Human DAPK1 Catalytic Subunit Complexed with Compound MW01-30-047SRM; X-ray diffraction 1.35Å
Protein #1 293 residues (96% resolved)

TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKESLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKPKDTQQALSSAWSHPQFE

TVFRQENVDDYYDTGEELGSGQFAVVKKCREKSTGLQYAAKFIKKRRTKSSRRGVSREDIEREVSILKEIQHPNVITLHEVYENKTDVILILELVAGGELFDFLAEKESLTEEEATEFLKQILNGVYYLHSLQIAHFDLKPENIMLLDRNVPKPRIKIIDFGLAHKIDFGNEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANVSAVNYEFEDEYFSNTSALAKDFIRRLLVKDPKKRMTIQDSLQHPWIKPKDTQQALSSAWSHPQFE
Non polymer #2 A1BVM

InChI=1S/C18H18N6/c1-5-19-6-2-15(1)16-13-18(22-21-14-16)24-11-9-23(10-12-24)17-3-7-20-8-4-17/h1-8,13-14H,9-12H2

c1cnccc1c2cc(nnc2)N3CCN(CC3)c4ccncc4
Download coordinates
Reference