2025-03-29_00000399|ligand|9HHC

Crystal Structure of the Plasmodium falciparum Bromodomain PfBDP1 in complex with MPM2; X-ray diffraction 1.56Å
Protein #1 137 residues (94% resolved)

GPLGSPEFMNKQWYLLANQLILSLSKYEGGHIFEKLVDAKKQNCPDYYDVIKNPMSFSCIKTKLKKGQYAYPSEFVKDVQLIFDNCSLYNTSNSVVAITGKNIETYFNNQLIVMGYNNFILKEKKINDMLKLVEEEN

GPLGSPEFMNKQWYLLANQLILSLSKYEGGHIFEKLVDAKKQNCPDYYDVIKNPMSFSCIKTKLKKGQYAYPSEFVKDVQLIFDNCSLYNTSNSVVAITGKNIETYFNNQLIVMGYNNFILKEKKINDMLKLVEEEN
Non polymer #2 BU3

InChI=1S/C4H10O2/c1-3(5)4(2)6/h3-6H,1-2H3/t3-,4-/m1/s1

C[C@H]([C@@H](C)O)O
Non polymer #3 I5K

InChI=1S/C16H18N2O/c1-10-15-13(7-2-3-8-14(15)19)16(18-10)11-5-4-6-12(17)9-11/h4-6,9,18H,2-3,7-8,17H2,1H3

Cc1c2c(c([nH]1)c3cccc(c3)N)CCCCC2=O
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Reference