2025-03-22_00000243
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ligand
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9FDC
Co-crystal structure of Galectin-3 with an inhibitor;
X-ray diffraction 1.78Å
Protein #1
138 residues (100% resolved)
Raw Sequence ...
PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI
Canonical Sequence ...
PLIVPYNLPLPGGVVPRMLITILGTVKPNANRIALDFQRGNDVAFHFNPRFNENNRRVIVCNTKLDNNWGREERQSVFPFESGKPFKIQVLVEPDHFKVAVNDAHLLQYNHRVKKLNEISKLGISGDIDLTSASYTMI
Non polymer #2
2PE
InChI=1S/C18H38O10/c19-1-3-21-5-7-23-9-11-25-13-15-27-17-18-28-16-14-26-12-10-24-8-6-22-4-2-20/h19-20H,1-18H2
InChI=1S/C18H38O10/c19-1-3-21-5-7-23-9-11-25-13-15-27-17-18-28-16-14-26-12-10-24-8-6-22-4-2-20/h19-20H,1-18H2
SMILES: C(COCCOCCOCCOCCOCCOCCOCCOCCO)O
C(COCCOCCOCCOCCOCCOCCOCCOCCO)O
Non polymer #3
A1IB4
InChI=1S/C22H19Cl2F3N4O5/c1-30(12-5-10(23)4-11(24)6-12)22(35)21-20(34)18(19(33)16(8-32)36-21)31-7-15(28-29-31)9-2-13(25)17(27)14(26)3-9/h2-7,16,18-21,32-34H,8H2,1H3/t16-,18+,19+,20-,21-/m1/s1
InChI=1S/C22H19Cl2F3N4O5/c1-30(12-5-10(23)4-11(24)6-12)22(35)21-20(34)18(19(33)16(8-32)36-21)31-7-15(28-29-31)9-2-13(25)17(27)14(26)3-9/h2-7,16,18-21,32-34H,8H2,1H3/t16-,18+,19+,20-,21-/m1/s1
SMILES: CN(c1cc(cc(c1)Cl)Cl)C(=O)[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)CO)O)n3cc(nn3)c4cc(c(c(c4)F)F)F)O
CN(c1cc(cc(c1)Cl)Cl)C(=O)[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)CO)O)n3cc(nn3)c4cc(c(c(c4)F)F)F)O
Non polymer #4
SCN
InChI=1S/CHNS/c2-1-3/h3H/p-1
InChI=1S/CHNS/c2-1-3/h3H/p-1
SMILES: C(#N)[S-]
C(#N)[S-]
Biounit #1
monomer
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Model
Reference
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