2025-03-01_00000017
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ligand
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7H6I
THE 2.10 A CRYSTAL STRUCTURE OF HUMAN CHYMASE IN COMPLEX WITH 5-fluoro-3-(methanesulfonamidomethyl)-1-(naphthalen-1-ylmethyl)indole-2-carboxylic acid;
X-ray diffraction 2.10Å
Protein #1
226 residues (97% resolved)
Raw Sequence ...
IIGGTESKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFPSQKNFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGVAQGIVSYGRSDAKPPAVFTRISHYRPWINQILQAN
Canonical Sequence ...
IIGGTESKPHSRPYMAYLEIVTSNGPSKFCGGFLIRRNFVLTAAHCAGRSITVTLGAHNITEEEDTWQKLEVIKQFRHPKYNTSTLHHDIMLLKLKEKASLTLAVGTLPFPSQKNFVPPGRMCRVAGWGRTGVLKPGSDTLQEVKLRLMDPQACSHFRDFDHNLQLCVGNPRKTKSAFKGDSGGPLLCAGVAQGIVSYGRSDAKPPAVFTRISHYRPWINQILQAN
Non polymer #2
A1AO7
InChI=1S/C22H19FN2O4S/c1-30(28,29)24-12-19-18-11-16(23)9-10-20(18)25(21(19)22(26)27)13-15-7-4-6-14-5-2-3-8-17(14)15/h2-11,24H,12-13H2,1H3,(H,26,27)
InChI=1S/C22H19FN2O4S/c1-30(28,29)24-12-19-18-11-16(23)9-10-20(18)25(21(19)22(26)27)13-15-7-4-6-14-5-2-3-8-17(14)15/h2-11,24H,12-13H2,1H3,(H,26,27)
SMILES: CS(=O)(=O)NCc1c2cc(ccc2n(c1C(=O)O)Cc3cccc4c3cccc4)F
CS(=O)(=O)NCc1c2cc(ccc2n(c1C(=O)O)Cc3cccc4c3cccc4)F
Non polymer #3
ZN
InChI=1S/Zn/q+2
InChI=1S/Zn/q+2
SMILES: [Zn+2]
[Zn+2]
Biounit #1
monomer
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Model
Reference
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