2025-02-22_00000118
|
ligand
|
7HWJ
Group deposition of Coxsackievirus A16 (G-10) 2A protease in complex with inhibitors from the ASAP AViDD centre -- Crystal structure of Coxsackievirus A16 (G-10) 2A protease in complex with ASAP-0034457-001 (A71EV2A-x3944);
X-ray diffraction 1.37Å
Protein #1
144 residues (97% resolved)
Raw Sequence ...
SGAIYVGNYRVVNRHLATHNDWANLVWEDSSRDLLVSSTTAQGCDTIARCDCQTGVYYCSSRRKHYPVSFSKPSLIFVEASEYYPARYQSHLMLAVGHSEPGDCGGILRCQHGVVGIVSTGGNGLVGFADVRDLLWLDEEAMEQ
Canonical Sequence ...
SGAIYVGNYRVVNRHLATHNDWANLVWEDSSRDLLVSSTTAQGCDTIARCDCQTGVYYCSSRRKHYPVSFSKPSLIFVEASEYYPARYQSHLMLAVGHSEPGDCGGILRCQHGVVGIVSTGGNGLVGFADVRDLLWLDEEAMEQ
Non polymer #2
A1BN3
InChI=1S/C21H29N3O3/c1-2-23(13-15-8-9-15)21(27)17-6-3-5-16(11-17)12-19(25)24-10-4-7-18(14-24)20(22)26/h3,5-6,11,15,18H,2,4,7-10,12-14H2,1H3,(H2,22,26)/t18-/m0/s1
InChI=1S/C21H29N3O3/c1-2-23(13-15-8-9-15)21(27)17-6-3-5-16(11-17)12-19(25)24-10-4-7-18(14-24)20(22)26/h3,5-6,11,15,18H,2,4,7-10,12-14H2,1H3,(H2,22,26)/t18-/m0/s1
SMILES: CCN(CC1CC1)C(=O)c2cccc(c2)CC(=O)N3CCC[C@@H](C3)C(=O)N
CCN(CC1CC1)C(=O)c2cccc(c2)CC(=O)N3CCC[C@@H](C3)C(=O)N
Non polymer #3
DMS
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
SMILES: CS(=O)C
CS(=O)C
Non polymer #4
ZN
InChI=1S/Zn/q+2
InChI=1S/Zn/q+2
SMILES: [Zn+2]
[Zn+2]
Biounit #1
monomer
Download coordinates
Tube
Model
Reference
100%