2025-02-22_00000044
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ligand
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7HPG
PanDDA analysis group deposition -- Crystal Structure of ZIKV NS2B-NS3 protease in complex with ASAP-0015487-001;
X-ray diffraction 1.66Å
Protein #1
46 residues (85% resolved)
Raw Sequence ...
SMGKSVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLVEE
Canonical Sequence ...
SMGKSVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLVEE
Protein #2
168 residues (92% resolved)
Raw Sequence ...
MKEVKKGETTDGVYRVMTRRLLGSTQVGVGVMQEGVFHTMWHVTKGAALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGLSEVQLLAVPPGERAKNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQGKREEETPVE
Canonical Sequence ...
MKEVKKGETTDGVYRVMTRRLLGSTQVGVGVMQEGVFHTMWHVTKGAALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGLSEVQLLAVPPGERAKNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQGKREEETPVE
Non polymer #3
A1BGT
InChI=1S/C17H20N4O2/c1-12-9-18-7-5-15(12)20-16(22)14-3-2-8-21(17(14)23)11-13-4-6-19-10-13/h2-3,5,7-9,13,19H,4,6,10-11H2,1H3,(H,18,20,22)/t13-/m1/s1
InChI=1S/C17H20N4O2/c1-12-9-18-7-5-15(12)20-16(22)14-3-2-8-21(17(14)23)11-13-4-6-19-10-13/h2-3,5,7-9,13,19H,4,6,10-11H2,1H3,(H,18,20,22)/t13-/m1/s1
SMILES: Cc1cnccc1NC(=O)C2=CC=CN(C2=O)C[C@@H]3CCNC3
Cc1cnccc1NC(=O)C2=CC=CN(C2=O)C[C@@H]3CCNC3
Non polymer #4
DMS
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
SMILES: CS(=O)C
CS(=O)C
Biounit #1
hetero-1-1-mer
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Model
Reference
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