2025-02-22_00000037
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ligand
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7HP9
PanDDA analysis group deposition -- Crystal Structure of ZIKV NS2B-NS3 protease in complex with ASAP-0015097-001;
X-ray diffraction 2.16Å
Protein #1
46 residues (85% resolved)
Raw Sequence ...
SMGKSVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLVEE
Canonical Sequence ...
SMGKSVDMYIERAGDITWEKDAEVTGNSPRLDVALDESGDFSLVEE
Protein #2
168 residues (93% resolved)
Raw Sequence ...
MKEVKKGETTDGVYRVMTRRLLGSTQVGVGVMQEGVFHTMWHVTKGAALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGLSEVQLLAVPPGERAKNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQGKREEETPVE
Canonical Sequence ...
MKEVKKGETTDGVYRVMTRRLLGSTQVGVGVMQEGVFHTMWHVTKGAALRSGEGRLDPYWGDVKQDLVSYCGPWKLDAAWDGLSEVQLLAVPPGERAKNIQTLPGIFKTKDGDIGAVALDYPAGTSGSPILDKCGRVIGLYGNGVVIKNGSYVSAITQGKREEETPVE
Non polymer #3
A1BGP
InChI=1S/C18H22N4OS/c23-18(16-12-24-17(21-16)14-4-2-7-20-10-14)22-8-5-15(11-22)13-3-1-6-19-9-13/h1,3,6,9,12,14-15,20H,2,4-5,7-8,10-11H2
InChI=1S/C18H22N4OS/c23-18(16-12-24-17(21-16)14-4-2-7-20-10-14)22-8-5-15(11-22)13-3-1-6-19-9-13/h1,3,6,9,12,14-15,20H,2,4-5,7-8,10-11H2
SMILES: c1cc(cnc1)[C@H]2CCN(C2)C(=O)c3csc(n3)[C@H]4CCCNC4
c1cc(cnc1)[C@H]2CCN(C2)C(=O)c3csc(n3)[C@H]4CCCNC4
Non polymer #4
DMS
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
InChI=1S/C2H6OS/c1-4(2)3/h1-2H3
SMILES: CS(=O)C
CS(=O)C
Biounit #1
hetero-1-1-mer
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Model
Reference
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