2025-01-18_00000334|medium|9J0C

Site-Specific Introduction of Sulfoxides and Sulfones into Polyketide Scaffold through a Relayed Chemo-Biosynthetic Strategy; X-ray diffraction 1.60Å
Protein #1 529 residues (95% resolved)

GSHMTATENADGRTRRRLDELARRRAELAAQATERGAGRQHAKGKLTARERIDLLLDPDSFTELDALARHRCHNYGMEEQRPYGDGVVTGYGTIDGRKVCVYAQDFTVLGGSLGEVFGEKIIKVLDLAIRTGCPVIGINDSGGARIQEGVVSLAYYAELVKRHVAASGVIPQISLIIGPCAGGAVYAPATTDLVVMVEDISHMFVTGPDVLQAVTGQTVGMEELGGAHRHNAVSGAAHYMAADEKDAFDYVRMVLGHLPSNNMGDTPVFAPTAARELTEADRALDTLIPDRTAESYDMMRVVNAVIDDGELTQFHQLFAPNVICGLARVEGHSVGVVANQPTHLAGALDIDASEKAARFIRFCDAFHVPVLTFVDVPGFLTSMEQERDGIIRRGAKLIYAYCEATVPMVTVITRKAYGGGYGVMGSKHLGIDVNLAWPTAEIAVMGGESAVRIIHRQDIRQAEDPEETRERLVSEYTETMCTPYVAAERGYVDAVIMPHETRAQVATALDTLRDKRMTRLPRKHGNIPL

GSHMTATENADGRTRRRLDELARRRAELAAQATERGAGRQHAKGKLTARERIDLLLDPDSFTELDALARHRCHNYGMEEQRPYGDGVVTGYGTIDGRKVCVYAQDFTVLGGSLGEVFGEKIIKVLDLAIRTGCPVIGINDSGGARIQEGVVSLAYYAELVKRHVAASGVIPQISLIIGPCAGGAVYAPATTDLVVMVEDISHMFVTGPDVLQAVTGQTVGMEELGGAHRHNAVSGAAHYMAADEKDAFDYVRMVLGHLPSNNMGDTPVFAPTAARELTEADRALDTLIPDRTAESYDMMRVVNAVIDDGELTQFHQLFAPNVICGLARVEGHSVGVVANQPTHLAGALDIDASEKAARFIRFCDAFHVPVLTFVDVPGFLTSMEQERDGIIRRGAKLIYAYCEATVPMVTVITRKAYGGGYGVMGSKHLGIDVNLAWPTAEIAVMGGESAVRIIHRQDIRQAEDPEETRERLVSEYTETMCTPYVAAERGYVDAVIMPHETRAQVATALDTLRDKRMTRLPRKHGNIPL
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Reference