2025-01-18_00000194
|
ligand
|
9DNV
SARS-CoV-2 papain-like protease (PLpro) with inhibitor Jun13308;
X-ray diffraction 2.40Å
Protein #1
318 residues (97% resolved)
Raw Sequence ...
SNAEVRTIKVFTTVDNINLHTQVVDMSMTYGQQFGPTYLDGADVTKIKPHNSHEGKTFYVLPNDDTLRVEAFEYYHTTDPSFLGRYMSALNHTKKWKYPQVNGLTSIKWADNNCYLATALLTLQQIELKFNPPALQDAYYRARAGEAANFCALILAYCNKTVGELGDVRETMSYLFQHANLDSCKRVLNVVCKTCGQQQTTLKGVEAVMYMGTLSYEQFKKGVQIPCTCGKQATKYLVQQESPFVMMSAPPAQYELKHGTFTCASEYTGNYQCGHYKHITSKETLYCIDGALLTKSSEYKGPITDVFYKENSYTTTIK
Canonical Sequence ...
SNAEVRTIKVFTTVDNINLHTQVVDMSMTYGQQFGPTYLDGADVTKIKPHNSHEGKTFYVLPNDDTLRVEAFEYYHTTDPSFLGRYMSALNHTKKWKYPQVNGLTSIKWADNNCYLATALLTLQQIELKFNPPALQDAYYRARAGEAANFCALILAYCNKTVGELGDVRETMSYLFQHANLDSCKRVLNVVCKTCGQQQTTLKGVEAVMYMGTLSYEQFKKGVQIPCTCGKQATKYLVQQESPFVMMSAPPAQYELKHGTFTCASEYTGNYQCGHYKHITSKETLYCIDGALLTKSSEYKGPITDVFYKENSYTTTIK
Non polymer #2
A1BEH
InChI=1S/C29H32N6O/c1-18-9-10-21(35-17-22-11-23(35)16-33(22)3)12-25(18)29(36)31-19(2)26-13-28(20-14-30-34(4)15-20)32-27-8-6-5-7-24(26)27/h5-10,12-15,19,22-23H,11,16-17H2,1-4H3,(H,31,36)
InChI=1S/C29H32N6O/c1-18-9-10-21(35-17-22-11-23(35)16-33(22)3)12-25(18)29(36)31-19(2)26-13-28(20-14-30-34(4)15-20)32-27-8-6-5-7-24(26)27/h5-10,12-15,19,22-23H,11,16-17H2,1-4H3,(H,31,36)
SMILES: Cc1ccc(cc1C(=O)N[C@H](C)c2cc(nc3c2cccc3)c4cnn(c4)C)N5C[C@H]6C[C@@H]5CN6C
Cc1ccc(cc1C(=O)N[C@H](C)c2cc(nc3c2cccc3)c4cnn(c4)C)N5C[C@H]6C[C@@H]5CN6C
Non polymer #3
ACY
InChI=1S/C2H4O2/c1-2(3)4/h1H3,(H,3,4)
InChI=1S/C2H4O2/c1-2(3)4/h1H3,(H,3,4)
SMILES: CC(=O)O
CC(=O)O
Non polymer #4
CL
InChI=1S/ClH/h1H/p-1
InChI=1S/ClH/h1H/p-1
SMILES: [Cl-]
[Cl-]
Non polymer #5
ZN
InChI=1S/Zn/q+2
InChI=1S/Zn/q+2
SMILES: [Zn+2]
[Zn+2]
Biounit #1
monomer
Download coordinates
Tube
Model
Reference
100%