2024-11-02_00000390|ligand|9JQI

Crystal structure of calmodulin in complex with KN93 (1:1 complex); X-ray diffraction 2.10Å
Protein #1 155 residues (93% resolved)

GPH(MSE)ADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTV(MSE)RSLGQNPTEAELQD(MSE)INEVDADGNGTIDFPEFLT(MSE)(MSE)ARK(MSE)KDTDSEEEIREAFRVFDKDGNGYISAAELRHV(MSE)TNLGEKLTDEEVDE(MSE)IREADIDGDGQVNYEEFVQ(MSE)(MSE)TAKNGL

GPHMADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTAKNGL
Non polymer #2 CA

InChI=1S/Ca/q+2

[Ca+2]
Non polymer #3 KN9

InChI=1S/C26H29ClN2O4S/c1-28(17-5-6-21-9-11-23(27)12-10-21)20-22-7-3-4-8-26(22)29(18-19-30)34(31,32)25-15-13-24(33-2)14-16-25/h3-16,30H,17-20H2,1-2H3/b6-5+

CN(C/C=C/c1ccc(cc1)Cl)Cc2ccccc2N(CCO)S(=O)(=O)c3ccc(cc3)OC
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Reference