2024-11-02_00000363|medium|9GKV

Crystal Structure of Deacetylase (HdaH) from Vibrio cholerae in complex with SAHA; X-ray diffraction 1.90Å
Protein #1 318 residues (97% resolved)

MAHHHHHHVGTMIPLIYHPIYSQLDLPVGHRYPINKYRLLYEEIVRQREQSEAWQASFEFHTPIAAELSRITPLHDPDYVQALLEGRLPAAKMRRIGFPWSKTLIERTLHSVGGTCLTVEQALQSGVAIHLSGGYHHAHADFGSGFCLFNDLAIAAHFALSLPSVDKVLIIDSDVHHGDGTATLCAERDDIITLSFHCDKNFPARKPASSMDVGFANQTGDEEFLSTFIQVVEMAVNLHRPDLILYDAGVDIHNDDELGYLSISQAAIAQRDRFMLGLAKQESIPIACVIGGGYREDHAALVPLHLELLKAALLSAGY

MAHHHHHHVGTMIPLIYHPIYSQLDLPVGHRYPINKYRLLYEEIVRQREQSEAWQASFEFHTPIAAELSRITPLHDPDYVQALLEGRLPAAKMRRIGFPWSKTLIERTLHSVGGTCLTVEQALQSGVAIHLSGGYHHAHADFGSGFCLFNDLAIAAHFALSLPSVDKVLIIDSDVHHGDGTATLCAERDDIITLSFHCDKNFPARKPASSMDVGFANQTGDEEFLSTFIQVVEMAVNLHRPDLILYDAGVDIHNDDELGYLSISQAAIAQRDRFMLGLAKQESIPIACVIGGGYREDHAALVPLHLELLKAALLSAGY
Non polymer #2 ACT

InChI=1S/C2H4O2/c1-2(3)4/h1H3,(H,3,4)/p-1

CC(=O)[O-]
Non polymer #3 K

InChI=1S/K/q+1

[K+]
Non polymer #4 SHH

InChI=1S/C14H20N2O3/c17-13(15-12-8-4-3-5-9-12)10-6-1-2-7-11-14(18)16-19/h3-5,8-9,19H,1-2,6-7,10-11H2,(H,15,17)(H,16,18)

c1ccc(cc1)NC(=O)CCCCCCC(=O)NO
Non polymer #5 ZN

InChI=1S/Zn/q+2

[Zn+2]
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Reference