2024-10-05_00000119|medium|8Y58

Crystal structure of TRIM21 PRYSPRY (D355A) in complex with acepromazine.; X-ray diffraction 1.60Å
Protein #1 192 residues (95% resolved)

GPMVHITLDPDTANPWLILSEDRRQVRLGDTQQSIPGNEERFDSYPMVLGAQHFHSGKHYWEVDVTGKEAWALGVCRDSVRRKGHFLLSSKSGFWTIWLWNKQKYEAGTYPQTPLHLQVPPCQVGIFLDYEAGMVSFYNITDHGSLIYSFSECAFTGPLRPFFSPGFNDGGKNTAPLTLCPLNIGSQGSTDY

GPMVHITLDPDTANPWLILSEDRRQVRLGDTQQSIPGNEERFDSYPMVLGAQHFHSGKHYWEVDVTGKEAWALGVCRDSVRRKGHFLLSSKSGFWTIWLWNKQKYEAGTYPQTPLHLQVPPCQVGIFLDYEAGMVSFYNITDHGSLIYSFSECAFTGPLRPFFSPGFNDGGKNTAPLTLCPLNIGSQGSTDY
Non polymer #2 FMT

InChI=1S/CH2O2/c2-1-3/h1H,(H,2,3)

C(=O)O
Non polymer #3 PMZ

InChI=1S/C19H22N2OS/c1-14(22)15-9-10-19-17(13-15)21(12-6-11-20(2)3)16-7-4-5-8-18(16)23-19/h4-5,7-10,13H,6,11-12H2,1-3H3

CC(=O)c1ccc2c(c1)N(c3ccccc3S2)CCCN(C)C
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Reference