2024-05-11_00000285|ligand|8V9O

Imaging scaffold engineered to bind the therapeutic protein target BARD1; X-ray diffraction 3.81Å
Protein #1 178 residues (89% resolved)

MRITTKVGDKGSTRLFGGEEVWKDDPIIEANGTLDELTSFIGEAKHYVDEEMKGILEEIQNDIYKIMGEIGSKGKIEGISEERIKWLAGLIERYSEMVNKLSFVLPGGTLESAKLDVCRTIARRAERKVATVLREFGIGTLAAIYLALLSRLLFLLARVIEIEKNKLKEVRSHHHHHH

MRITTKVGDKGSTRLFGGEEVWKDDPIIEANGTLDELTSFIGEAKHYVDEEMKGILEEIQNDIYKIMGEIGSKGKIEGISEERIKWLAGLIERYSEMVNKLSFVLPGGTLESAKLDVCRTIARRAERKVATVLREFGIGTLAAIYLALLSRLLFLLARVIEIEKNKLKEVRSHHHHHH
Protein #2 322 residues (93% resolved)

MFTRRGDQGETDLANRARVGKDSPVVEVQGTIDELNSFIGYALVLSRWDDIRNDLFRIQNDLFVLGEDVSTGGKGRTVTMDMIIYLIKRSVEMKAEIGKIELFVVPGGSVESASLHMARAVSRRLERRIKAASELTEINANVLLYANMLSNILFMHALISNKRKEELDKKLLEAARAGQDDEVAALLAKGADVNASDYKGTTPLHVAAWNGHLEIVDVLLARGADINASDSYGDTPLHLAANYGHLEIVDLLLRWGADVNASDSSGKTPLHLAAQDGHLEIVDVLLAHGADVNAQDKFGKTPFDLAIDNGNEDIAEVLQKAA

MFTRRGDQGETDLANRARVGKDSPVVEVQGTIDELNSFIGYALVLSRWDDIRNDLFRIQNDLFVLGEDVSTGGKGRTVTMDMIIYLIKRSVEMKAEIGKIELFVVPGGSVESASLHMARAVSRRLERRIKAASELTEINANVLLYANMLSNILFMHALISNKRKEELDKKLLEAARAGQDDEVAALLAKGADVNASDYKGTTPLHVAAWNGHLEIVDVLLARGADINASDSYGDTPLHLAANYGHLEIVDLLLRWGADVNASDSSGKTPLHLAAQDGHLEIVDVLLAHGADVNAQDKFGKTPFDLAIDNGNEDIAEVLQKAA
Non polymer #3 CA

InChI=1S/Ca/q+2

[Ca+2]
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Reference